| [1] |
Sun Y,Takada K,Takemoto Y,et al.Gliotoxin analogues from a marine-derived fungus,Penicilliumsp.,and their cytotoxic and histone methyltransferase inhibitory activities[J].J Nat Prod,2012,75(1):111-114.
|
| [2] |
Raju R,Piggott AM,Huang XC,et al.Nocardioazines:a novel bridged diketopiperazine scaffold from a marine-derived bacterium inhibits P-glycoprotein[J].Org Lett,2011,13(10):2770-2773.
|
| [3] |
Liao SR,Qin XC,Li D,et al.Design and synthesis of novel soluble 2,5-diketopiperazine derivatives as potential anticancer agents[J].Eur J Med Chem,2014,83:236-244.
|
| [4] |
Yamazaki Y,Tanaka K,Nicholson B,et al.Synthesis and structure-activity relationship study of antimicrotubule agents phenylahistin derivatives with a didehydropiperazine-2,5-dione structure[J].J Med Chem,2012,55(3):1056-1071.
|
| [5] |
Yamazaki Y,Sumikura M,Masuda Y,et al.Synthesis and structure-activity relationships of benzophenone-bearing diketopiperazine-type anti-microtubule agents[J].Bioorg Med Chem,2012,20(14):4279-4289.
|
| [6] |
El-Gendy BD,Rateb ME.Antibacterial activity of diketopiperazines isolated from a marine fungus using t-butoxycarbonyl group as a simple tool for purification[J].Bioorg Med Chem Lett,2015,25(16):3125-3128.
|
| [7] |
Liao SR,Xu Y,Tang Y,et al.Design,synthesis and biological evaluation of soluble 2,5-diketopiperazines derivatives as potential antifouling agents[J].RSC Adv,2015,5(63):51020-51026.
|
| [8] |
Sinha S,Srivastava R,Singh R,et al.Synthesis and antiviral properties of arabino and ribonucleosides of 1,3-dideazaadenine,4-nitro-1,3-dideazaadenine and diketopiperazine[J].Nucleosides Nucleotides,2004,23(12):1815-1824.
|
| [9] |
Borthwick AD, Liddle J, Davies DE, et al. Pyridyl-2,5-diketopiperazines as potent,selective,and orally bioavailable oxytocin antagonists:synthesis,pharmacokinetics,and in vivo potency[J].J Med Chem,2012,55(2):783-796.
|
| [10] |
Borthwick AD. 2, 5-Diketopiperazines: synthesis, reactions,medicinal chemistry,and bioactive natural products[J].Chem Rev,2012,112(7):3641-3716.
|
| [11] |
Yamazaki Y,Mori Y,Oda A,et al.Acid catalyzed monodehydro-2,5-diketopiperazine formation from N-α-ketoacyl amino acid amides[J].Tetrahedron,2009,65(18):3688-3694.
|
| [12] |
Ressurreição ASM,Delatouche R,Gennari C,et al.Bifunctional 2,5-diketopiperazines as rigid three-dimensional scaffolds in receptors and peptidomimetics[J].Eur J Org Chem,2011,2011(2):217-228.
|
| [13] |
Du YM,Creighton CJ,Reitz AB,et al.Noncovalent self-assembly of bicyclo[4.2.2] diketopiperazines:influence of Saturation in the bridging carbacyclic ring[J].Org Lett,2004,6(3):309-312.
|
| [14] |
Weatherhead-Kloster RA,Selby HD,Mash EA,et al.Organic crystal engineering with 1,4-piperazine-2,5-diones.6.Studies of the hydrogen-bond association of cyclo[(2-methylamino-4,7-dimethoxyindan-2-carboxylic acid)(2-amino-4,7-dimethoxyindan -2-carboxylic acid)][J].J Org Chem,2005,70(22):8693-8702.
|
| [15] |
Gillis EP,Eastman KJ,Hill MD,et al.Applications of fluorine in medicinal chemistry[J].J Med Chem,2015,58(21):8315-8359.
|
| [16] |
Yan Q,Wu SM,Ni LL,et al.Synthesis and antitumor activity of C-3 thiazolo[3,2-b][1,2,4] triazole-substituted pefloxacin derivatives[J].J China Pharm Univ(中国药科大学学报),2015,46(5):283-284.
|
| [17] |
Gao LZ,Xie YS,Hu GQ,et al.Synthesis,antibacterial and antitumor activities of 1-cycloproyl-6-fluoro-7-(hydrazone)-quinolin-4(1H)-one-carboxylic acids[J].J China Pharm Univ(中国药科大学学报),2014,45(6):662-664.
|
| [18] |
Li JS,Liao SR,Tang Y,et al.Synthesis and cytotoxic activities of 2,5-diketopiperazine derivatives by one-pot method[J].Chin J Synth Chem(合成化学),2015,12(23):1095-1099.
|
下载:
