某些阿朴菲类生物碱及其氧化,去氢衍生物对M—胆碱受体的作用
EFFECTS OF SOME APORPHINES AND THEIR OXIGENATED, DEHYDROGENATED DERIVATIVES ON M-CHOLINERGIC RECEPTORS
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摘要: 某些双苄基异喹啉及原小檗碱等异喹啉生物碱对M-胆碱受体有较高的亲和力,如粉防已碱Ki为7.3×10~(-8)mol/L。阿朴菲类生物碱亦属异喹啉类生物碱。此类生物碱有阿朴菲原
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Keywords:
- Oxocrebamine /
- Dicentrine /
- Dehydrocrebamine /
- Dehydrodicentrine /
- Oxidation state /
- M-Cholinergic receptor
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