Citation: | SONG Lin, WANG Mao, WEN Aidong, YANG Lin, JIA Yuntao, XIE Huiru, JIANG Xuehua, WANG Ling. Determination of agomelatine in human plasma by LC-MS/MS:application to a pharmacokinetic study in Chinese volunteers[J]. Journal of China Pharmaceutical University, 2014, 45(6): 698-702. DOI: 10.11665/j.issn.1000-5048.20140615 |
[1] |
Wang X, Ma HM, Zhou YS. The graphical synthetic routes of agomelatine[J].Chin J Med Chem(中国药物化学杂志),2012,99(4):334-336.
|
[2] |
Landolt HP,Wehrle R.Antagonism of serotonergic 5-HT2A/2C receptors:mutual improvement of sleep,cognition and mood[J].Eur J Neurosci,2009,29(9):1 795-1 809.
|
[3] |
Howland RH.Critical appraisal and update on the clinical utility of agomelatine,a melatonergic agonist,for the treatment of major depressive disease in adults[J].Neuropsychiatr Dis Treat,2009,5:563-576.
|
[4] |
Millan M,Gobert A,Lejeune F,et al.The novel melatonin agonist agomelatine(S20098)is an antagonist at 5-hydroxytryptamine 2C receptors,blockade of which enhances the activity of frontocortical dopaminergic and adrenergic pathways[J].J Pharmacol Exp Ther,2003,306(3):954-964.
|
[5] |
Banasr M,Soumier A,Hery M,et al.Agomelatine,a new antidepressant,induces regional changes in hippocampal neurogenesis[J].Biol Psychiatry,2006,59(11):1 087-1 096.
|
[6] |
Wei MJ,Zhang ZF,Zhang ZF.Discussion on accuracy in the analysis of biological samples and improvement measures[EB/OL].(2012-04-11)[2012-09-30] .http://www.cde.org.cn/dzkw.do?method=largePage&id=312642.
|
[7] |
European Medicines Agency. CHMP ASSESSMENT REPORT FOR Valdoxan[EB/OL].(2008-11-20)[2011-12-12] .http://www.ema.europa.eu/docs/en_GB/document_library/EPAR_-_Public_assessment_report/human/000915/WC500046226.pdf.
|
[8] |
European Medicines Agency.Guideline on the investigation of bioequivalence[EB/OL].(2010-01-20)[2011-12-12] .http://www.ema.europa.eu/docs/en_GB/document_library/Scientific_guideline/2010/01/WC500070039.pdf.
|
[9] |
Chow SC,Liu J.Design and Analysis of Bioavailability and Bioequivalence Studies[M].CRC Press,2000.
|
[10] |
Patil SR,Nerurkar KK,Kalamkar AM,et al.Validated LC-MS/MS method for quantification of agomelatine in human plasma and its application in a pharmacokinetic study[J].J Mass Spectrom,2012,47(1):23-28.
|
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