Citation: | CAI Qilin, LI Wenxing, YAN Zhen, YIN Lifang. Prediction of the bioequivalence of different crystal forms of rifampicin based on physiologically based pharmacokinetic model[J]. Journal of China Pharmaceutical University, 2022, 53(2): 207-214. DOI: 10.11665/j.issn.1000-5048.20220211 |
[1] |
.J Occup Environ Med,2020,62(7):e355-e369.
|
[2] |
Yulug B,Hanoglu L,Ozansoy M,et al.Therapeutic role of rifampicin in Alzheimer''s disease[J].Psychiatry Clin Neurosci,2018,72(3):152-159.
|
[3] |
Allen FH.The Cambridge structural database:a quarter of a million crystal structures and rising[J].Acta Crystallogr B,2002,58(Pt3Pt1):380-388.
|
[4] |
Censi R, di Martino P.Polymorph impact on the bioavailability and stability of poorly soluble drugs[J].Molecules,2015,20(10):18759-18776.
|
[5] |
Guo LL.Investigation on polymorphs and crystallization process of rifampicin(利福平多晶型及其结晶过程研究)[D].Tianjin:Tianjin University,2018.
|
[6] |
Zhao P,Zhang L,Grillo JA,et al.Applications of physiologically based pharmacokinetic (PBPK) modeling and simulation during regulatory review[J].Clin Pharmacol Ther,2011,89(2):259-267.
|
[7] |
Poggesi I,Snoeys J,van Peer A.The successes and failures of physiologically based pharmacokinetic modeling:there is room for improvement[J].Expert Opin Drug Metab Toxicol,2014,10(5):631-635.
|
[8] |
Agoram B,Woltosz WS,Bolger MB.Predicting the impact of physiological and biochemical processes on oral drug bioavailability[J].Adv Drug Deliv Rev,2001,50(
|
[9] |
U.S. Department of Health and Human Services Food and Drug Administration Center for Drug Evaluation and Research (CDER):Clinical drug interaction studies -cytochrome P450 enzyme-and transporter-mediated drug interactions guidance for industry[EB/OL].U.S.Food and Drug Administration,2020[
|
[10] |
Amidon GL,Tsume Y.Oral product input to the GI tract: GIS an oral product performance technology[J].Front Chem Sci Eng,2017,11(4):516-520.
|
[11] |
de Pinho Pessoa Nogueira L,de Oliveira YS,de C Fonseca J,et al.Crystalline structure of the marketed form of rifampicin:a case of conformational and charge transfer polymorphism[J].J Mol Struct,2018,1155:260-266.
|
[12] |
Biganzoli E,Cavenaghi LA,Rossi R,et al.Use of a Caco-2 cell culture model for the characterization of intestinal absorption of antibiotics[J].Farmaco,1999,54(9):594-599.
|
[13] |
Toutain PL,Bousquet-Mélou A.Plasma clearance[J].J Vet Pharmacol Ther,2004,27(6):415-425.
|
[14] |
U.S.Food and Drug Administration.FDA approves RIFADIN? IV (rifampin for injection USP)[EB/OL].(
|
[15] |
Becker C,Dressman JB,Junginger HE,et al.Biowaiver monographs for immediate release solid oral dosage forms:Rifampicin[J].J Pharm Sci,2009,98(7):2252-2267.
|
1. |
周德军,王珂洋,郝婷,张钰滢,赵桂琴. 三氮唑香豆素的合成进展. 化学研究与应用. 2024(04): 696-703 .
![]() | |
2. |
李卓远,史佳慧,刘楠,薛玉涛,李婉倩,蒋治坤,周佳雨,刘晖,熊山. 香豆素衍生物的生物活性研究进展. 精细与专用化学品. 2024(06): 23-30 .
![]() |