Citation: | CHENG Keguang, CHU Xiangwu, LIU Guanyan, SU Chunhua, DENG Shengping, PAN Hongmei. Synthesis and antitumor activities of 3-substituted estradiol-pyrimidine derivatives[J]. Journal of China Pharmaceutical University, 2014, 45(1): 26-32. DOI: 10.11665/j.issn.1000-5048.20140104 |
[1] |
Wei W,Ge JP,Ma HQ,et al.The application of low-dose EMP in the treatment of prostate cancer[J].Chin Clin Oncol(临床肿瘤学杂志),2007,12(6):432-434.
|
[2] |
An FR,Cui L,Zhu DQ.Development of a pure antiestrogen fulvestrant[J].Chin J Clin Pharmacol(中国临床药理学杂志),2002,18(2):156-158.
|
[3] |
Blockeel C.Estradiol valerate pretreatment in GnRH-antagonist cycles[J].Reprod BioMed Online,2012,25(2):223-224.
|
[4] |
Peralta-Torres J,Ake-Lopez J,Centurion-Castro F,et al.Comparison of estradiol cypionate and estradiol benzoate effects on ovaric activity,estrus and ovulation on anestrus Bos indicus cows[J].J Anim Vet Adv,2010,9(3):466-470.
|
[5] |
Verenich S,Gerk PM.Therapeutic promises of 2-methoxyestradiol and its drug disposition challenges[J].Mol Pharm,2010,7(6):2 030-2 039.
|
[6] |
Sharma U,Marquis JC,Dinaut AN,et al.Design,synthesis,and evaluation of estradiol-linked genotoxicants as anti-cancer agents[J].Bioorg Med Chem Lett,2004,14(14):3 829-3 833.
|
[7] |
Gupta A,Saha P,Descoteaux C,et al.Design,synthesis and biological evaluation of estradiol-chlorambucil hybrids as anticancer agents[J].Bioorg Med Chem Lett,2010,20(5):1 614-1 618.
|
[8] |
Miyahara S,Miyakoshi H,Yokogawa T,et al.Discovery of a novel class of potent human deoxyuridine triphosphatase inhibitors remarkably enhancing the antitumor activity of thymidylate synthase inhibitors[J].J Med Chem,2012,55(7):2 970-2 980.
|
[9] |
Miyahara S,Miyakoshi H,Yokogawa T,et al.Discovery of highly potent human deoxyuridine triphosphatase inhibitors based on the conformation restriction strategy[J].J Med Chem,2012,55(11):5 483-5 496.
|
[10] |
Miyakoshi H,Miyahara S,Yokogawa T,et al.1,2,3-Triazole-containing uracil derivatives with excellent pharmacokinetics as a novel class of potent human deoxyuridine triphosphatase inhibitors[J].J Med Chem,2012,55(14):6 427-6 437.
|
[11] |
Mosmann T.Rapid colorimetric assay for cellular growth and survival:application to proliferation and cytotoxicity assays[J].J Immunol Methods,1983,65(1):55-63.
|
[1] | GAO Yuan, JIANG Kun, LI Li, XI Yi-feng. Bioavailability enhancement of baicalein by nanosuspension[J]. Journal of China Pharmaceutical University, 2011, 42(4): 314-318. |
[2] | Lü Wen-li, RONG Fei, PING Qi-neng. Preparation,dissolution and bioavailability of lycopene-Poloxamer 188 solid dispersion[J]. Journal of China Pharmaceutical University, 2009, 40(6): 514-518. |
[3] | CHEN Ling-ping, L Wen-li, PING Qi-neng. Preparation and bioavailability of bupropion hydrochloride sustained-release pellets[J]. Journal of China Pharmaceutical University, 2009, 40(5): 421-425. |
[4] | Pharmacokinetics and Relative Bioavailability of Gliquidone Capsules and Tablets[J]. Journal of China Pharmaceutical University, 2000, (6): 19-21. |
[5] | Study on the Preparation of Ibuprofen Granules and Determination of Their Bioavailability[J]. Journal of China Pharmaceutical University, 1999, (3): 23-26. |
[6] | Pharmacokinetics and Relative Bioavailability of Cyclosporin Pearls in Healthy Volunteers[J]. Journal of China Pharmaceutical University, 1996, (6): 20-22. |
[7] | Pharmacokinetics and Bioavailability of Ribavirin in 9 Chinese Healthy Volunteers[J]. Journal of China Pharmaceutical University, 1994, (6): 325-327. |
[8] | Relative Bioavailability and Bioequivalence Assessment of Domestic Amiloride Tablet[J]. Journal of China Pharmaceutical University, 1994, (1): 9-11. |
[9] | Dissolution Test in Vitro and Bioavailability Study on Sustained-Release Verapamil Hydrochloride Tablets[J]. Journal of China Pharmaceutical University, 1992, (2): 88-92. |
[10] | Lv Mingsheng, Wu Guangchen, Lv Zhenda, Yue Zhiwei. DETERMINATION OF THE RELATIVE BIOAVAILABILITY OF HYDROCHLOROTHIAZIDE TABLETS IN HUMAN[J]. Journal of China Pharmaceutical University, 1983, (1): 55-60. |