Citation: | MAO Zewei, WAN Chunping, ZHENG Xi, JIANG Yuan, RAO Gaoxiong. Synthesis and biological activities of novel hybrid compounds based on piperazines and acetophenones[J]. Journal of China Pharmaceutical University, 2014, 45(5): 517-521. DOI: 10.11665/j.issn.1000-5048.20140502 |
[1] |
Huang PL,Lu CM,Yen MH,et al.Acetophenones from Cynanchum taiwanianum[J].Phytochemistry,1995,40(2):537-541.
|
[2] |
Adsersen A,Smitt UW,Simonsen HT,et al.Prenylated acetophenones from Melicope obscura and Melicope obtusifolia ssp. obtusifolia var. arborea and their distribution in Rutaceae[J].Biochem Syst Ecol,2007,35(7):447-453.
|
[3] |
Lavault M,Richomme P,Bruneton J. Acetophenones and new pregnane glycosides from the roots of Vincetoxicum hirundinaria[J].Fitoterapia,1999,70(2):216-220.
|
[4] |
Jacob RG,Alves D.In vitro antioxidant activity and in vivo antidepressant-like effect of α-(phenylselanyl)acetophenone in mice[J].Pharmacol Biochem Behav,2012,102(1):21-29.
|
[5] |
Alang G,Kaur G,Kaur,R. Synthesis,characterization,and biological evaluation of certain 6-methyl-2(3H)-benzo-1,3-thiazolyl-1′-ethylidene-2-(o,p-substituted acetophenones)hydrazine analogs[J].J Young Pharm,2010,2(4):394-398.
|
[6] |
Dorsch W,Müller A,Christoffel V,et al.Antiasthmatic acetophenones -an in vivo study on structure activity relationship[J].Phytomedicine,1994,1(1):47-54.
|
[7] |
Singh A,Chisti Y,Banerjee UC,et al.Stereoselective biocatalytic hydride transfer to substituted acetophenones by the yeast Metschnikowia koreensis[J].Process Biochem,2012, 47(12):2 398-2 404.
|
[8] |
Chikhale RV,Bhole RP,Khedekar PB,et al.Synthesis and pharmacological investigation of 3-(substituted 1-phenylethanone)-4-(substituted phenyl)-1,2,3,4-tetrahydropyrimidine-5-carboxylates[J].Eur J Med Chem,2009,44(9):3 645-3 653.
|
[9] |
Zheng L,Li Y,Ge D,et al.Synthesis of novel oxime-containing pyrazole derivatives and discovery of regulators for apoptosis and autophagy in A549 lung cancer cells[J].Bioorg Med Chem Lett,2010,20(16):4 766-4 770.
|
[10] |
Zhang LR,Liu ZJ,Zhang H,et al.Synthesis,biological evaluation and molecular docking studies of novel 2-(1,3,4-oxadiazol-2-ylthio)-1-phenylethanone derivatives[J].Bioorg Med Chem,2012,20(11):3 615-3 621.
|
[11] |
Jason MN,Lee MB,Robert GB,et al.Catalytic C-O bond cleavage of 2-aryloxy-1-arylethanols and its application to the depolymerization of lignin-related polymers[J].J Am Chem Soc,2010,132(36):12 554-12 555.
|
[12] |
Ajay A,Singh V,Singh S,et al.Synthesis and bio-evaluation of alkylaminoaryl phenyl cyclopropyl methanones as antitubercular and antimalarial agents[J].Bioorg Med Chem,2010,18(23):8 289-8 301.
|
[13] |
Ge YQ,Cheng RB,Chen Z,et al.Cryptotanshinone induces cell cycle arrest and apoptosis of multidrug resistant human chronic myeloid leukemia cells by inhibiting the activity of eukaryotic initiation factor 4E[J].Mol Cell Biochem,2012,368(1):17-25.
|
[14] |
Langfied RD,Scarano FJ,Heitzman ME,et al.Use of a modified microplate bioassay method to investigate antibacterial activity in the Peruvian medicinal plant Peperomia galioides[J].J Ethnopharmacol,2004,94(2/3):279-281.
|
[15] |
Wang JJ,Zhao BY,Zhang WM,et al.Experimental study on antimicrobial effects of extracts from Astragalus strictus in vitro[J].Acta Agric Boreali-Occidentalis Sin(西北农业学报),2007,16(2):108-112.
|
[1] | LIU Li, LIU Zijin, TANG Jun, HE Guangwei, LIU Weizhong. Optimized synthesis process of tofacitinib citrate[J]. Journal of China Pharmaceutical University, 2022, 53(6): 685-689. DOI: 10.11665/j.issn.1000-5048.20220606 |
[2] | WU Xufeng, CHAI Shiying, LIU Jianhong, WANG Zhihui, YIN Ruifeng, CAO Ruiwei, SUN Xinqiang. Improvement of synthetic route of brivudine[J]. Journal of China Pharmaceutical University, 2022, 53(1): 41-45. DOI: 10.11665/j.issn.1000-5048.20220106 |
[3] | WANG Dong, ZHONG Jian, WANG Ling, ZHOU Zhihui, JIANG Haiting, LUO Peng, WANG Xizhi, WANG Chongyi. Improved synthetic process of apremilast[J]. Journal of China Pharmaceutical University, 2021, 52(5): 536-540. DOI: 10.11665/j.issn.1000-5048.20210504 |
[4] | HAN Chengqun, ZOU Qiaogen, SUN Qian, XIA Yunyan. Improvement of synthesis process of mirabegron[J]. Journal of China Pharmaceutical University, 2020, 51(4): 449-453. DOI: 10.11665/j.issn.1000-5048.20200409 |
[5] | ZHANG Qiuyue, YOU Qidong, YANG Jinpeng. Process improvement on the synthesis of atomoxetine[J]. Journal of China Pharmaceutical University, 2019, 50(4): 405-409. DOI: 10.11665/j.issn.1000-5048.20190404 |
[6] | LIU Li, WANG Chen, LIU Lixin, JI Tingting. Improved synthesis of analgesic pentazocine[J]. Journal of China Pharmaceutical University, 2018, 49(5): 568-571. DOI: 10.11665/j.issn.1000-5048.20180508 |
[7] | MA Li, ZHANG Menghan, XU Zhiwei, SUN Ying′ai, ZHU Jing, HUANG Yingbo, ZHANG Dayong. A new synthetic process of dapagliflozin[J]. Journal of China Pharmaceutical University, 2017, 48(1): 42-45. DOI: 10.11665/j.issn.1000-5048.20170106 |
[8] | WEI Qingjie, QIAO Junhua, CHEN Jianjun, GAO Zhigang, LI Yaqing. An improvement for synthesis of ceftriaxone sodium[J]. Journal of China Pharmaceutical University, 2016, 47(2): 163-165. DOI: 10.11665/j.issn.1000-5048.20160206 |
[9] | Improve on the Synthetic Process of Bezafibrate[J]. Journal of China Pharmaceutical University, 2003, (3): 80-81. |
[10] | Improved Process of Nimodipine[J]. Journal of China Pharmaceutical University, 1998, (3): 82-83. |