Advanced Search
Cao Mingzhu, Hu Shuchen, Li Minghua, Zhang Song. The Synthesis of Carboxylic Esters of Dihydroartemisinine[J]. Journal of China Pharmaceutical University, 1982, (1): 53-54.
Citation: Cao Mingzhu, Hu Shuchen, Li Minghua, Zhang Song. The Synthesis of Carboxylic Esters of Dihydroartemisinine[J]. Journal of China Pharmaceutical University, 1982, (1): 53-54.
shu

The Synthesis of Carboxylic Esters of Dihydroartemisinine

More Information
    Graphical Abstract
    • Abstract
  • Artemisinine is a new type of fast-acting suppresive antimalarial drug. Dihydroar-temisinine is its reduced product. We have prepared nine oarboxylio esters of dihvdroartemisinine for evaluation of their antimalarial potency. All the new compounds have been tested for suppressive antimalarial activity against p. herghei in mice, four Ⅰ、Ⅱ、Ⅲ、Ⅸ,) of them are superior to artemisinine.
    • FullText(HTML)
    • References (0)
    • Related Articles

  • Related Articles

    [1]MOU Yi, CHEN Tong, HUANG Zhangjian, LAI Yisheng, PENG Sixun, JI Hui, ZHANG Yihua. Design, synthesis and anti-inflammatory evaluation of CDDO-Me ester prodrugs[J]. Journal of China Pharmaceutical University, 2016, 47(6): 661-665. DOI: 10.11665/j.issn.1000-5048.20160605
    [2]WU Mingming, FANG Lei, GOU Shaohua, CHEN Li. 以2-甲基-2-取代苯氧基丙酸为离去基团的铂(Ⅱ)配合物的合成、表征及细胞毒活性[J]. Journal of China Pharmaceutical University, 2013, 44(4): 303-306. DOI: 10.11665/j.issn.1000-5048.20130403
    [3]WU Wen-chao, ZHANG Chi, SHEN Zu-cheng, CHEN Li-ping, CHEN Li-qin. Synthesis of deuterium-labeled losartan and losartan 5-carboxylic acid with improved isotopic enrichment[J]. Journal of China Pharmaceutical University, 2012, 43(6): 497-501.
    [4]XU Bei-hua, ZHOU Hui-yan. Synthesis and characterization of camptothecin-polyethylene glycol ester prodrugs[J]. Journal of China Pharmaceutical University, 2012, 43(2): 142-146.
    [5]A NewSimple Synthesis Method of the 1-Benzenemethyl Piperidine-4-Carboxylic Acid[J]. Journal of China Pharmaceutical University, 2000, (1): 5-6.
    [6]Synthesis of Dihydrobenzopyran-4-Oximes and Oxime Esters[J]. Journal of China Pharmaceutical University, 1995, (3): 129-133.
    [7]Synthesis of 7-Amino-3-Vinyl-3-Cephem-4-Carboxylic Acid[J]. Journal of China Pharmaceutical University, 1993, (4): 246-247.
    [8]SYNTHESIS OF OXIMINO ESTERS OF VANILLIN,VERATRALDEHYDE AND PIPERONAL[J]. Journal of China Pharmaceutical University, 1987, (1): 1-7.
    [9]SYNTHESIS OF 3-BROMOMETHYLCEPHEMBEN- ZHYDRYL ESTER S-OXIDE[J]. Journal of China Pharmaceutical University, 1985, (1): 4-6.
    [10]Shen Xinhua, Xu Fang, Liao Qingjiang. SYNTHESIS OF 3.3.5-TRIMETHYLCYCLOHEXANOL ESTERS[J]. Journal of China Pharmaceutical University, 1983, (2): 19-26.

  • Cited by

    Periodical cited type(1)

    1. 王莉婷，刘湉，母磊鑫，王凯赫，柯彩依，吉莉，徐广，马群. 基于网络药理学和分子对接技术探讨车前子治疗高尿酸血症的作用机制. 江苏大学学报(医学版). 2024(05): 369-376+382 .

    Other cited types(2)

Catalog

    Get Citation
    PDF
    XML
    Article views (1083) PDF downloads (772) Cited by(3)
    Turn off MathJax
    Article Contents
    Abstract
    Related Articles

    Copyright © Journal of China Pharmaceutical University苏ICP备12050101号-2

    Address：24 Tongjia Lane, Nanjing City, Jiangsu Province （210009）Tel: 025-83271566E-mail: xuebao@cpu.edu.cn

    Supported by: Beijing Renhe Information Technology Co., Ltd.  Baidu Analytics

    Total visits：457676

    /

    DownLoad:  Full-Size Img  PowerPoint
    Return
    Return